SCHEMBL7925071

SCHEMBL7925071

NC(=O)c1ccc(N)cc1N1CCC(Cc2ccccc2)CC1.Nc1ccc(C(=O)N2CCC(Cc3ccccc3)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA7 P43166 1/20 0.55
CA9 Q16790 1/20 0.55
CA14 Q9ULX7 1/20 0.55
HTT P42858 2/20 0.53
GAA P10253 1/20 0.50
CCR3 P51677 1/20 0.49
CYP2C9 P11712 3/20 0.48
CYP2C19 P33261 3/20 0.48
MAPK14 Q16539 3/20 0.48
HTR2B P41595 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 1/20 0.48
NPBWR1 P48145 1/20 0.48
MCHR1 Q99705 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7617666 0.91 MAPT (0.55) CA12CA1CA2CA9HTT
SCHEMBL7238944 0.85 CA12 (0.73) CA12CA1CA2CA7CA9
SCHEMBL10719972 0.79 HTT (0.78) CA12CA1CA2CA7CA9
SCHEMBL9058262 0.78 CA12 (0.63) CA12CA1CA2CA7CA9
SCHEMBL2729282 0.77 CYP2C9 (0.60) CA12CA1CA2CA7CA9
SCHEMBL5165728 0.77 GAA (0.65) CA12CA1CA2CA7CA9
SCHEMBL7232623 0.76 CYP2C9 (0.73) HTTCYP2C9CYP2C19MAPK14HTR2B
SCHEMBL7232379 0.76 HTT (0.73) CA12CA1CA2CA7CA9
SCHEMBL4731357 0.74 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL7238728 0.74 HTT (0.70) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107758-A2 USE OF PIPERIDINES AND/OR PIPERAZINES AS INHIBITORS OF P38-ALPHA KINASE SCIOS INC. (US) 2001-06-20 EP disclosed
WO-2000012074-A2 USE OF PIPERIDINES AND/OR PIPERAZINES AS INHIBITORS OF P38-ALPHA KINASE SCIOS INC. (US) 2000-03-09 WO disclosed