SCHEMBL7925156

SCHEMBL7925156

Bc1ccc2ccc(B)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
CYP2A6 P11509 1/20 0.40
APEX1 P27695 2/20 0.35
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14304431 0.89 CYP2A6 (0.37) CYP1A2CYP2A6
SCHEMBL319839 0.84 CYP2A6 (0.48) CYP1A2CYP2A6ESR1ESR2
SCHEMBL24808500 0.84 CYP2A6 (0.54) CYP2A6
SCHEMBL21215460 0.84 CYP2A6 (0.54) CYP1A2CYP2A6
SCHEMBL14733926 0.84 CYP1A2 (0.54) CYP1A2ESR1ESR2
SCHEMBL11959837 0.82 ALDH1A1 (0.50) CYP1A2CYP2A6
SCHEMBL14983311 0.82 ALDH1A1 (0.50) CYP1A2CYP2A6
SCHEMBL12809407 0.80 ALDH1A1 (0.39) CYP1A2CYP2A6
SCHEMBL22705421 0.78 HPRT1 (0.41) CYP1A2CYP2A6
SCHEMBL13865663 0.76 CYP2A6 (0.52) CYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499115-B1 PROCESS FOR PREPARING HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB HOLDINGS IRELAND (CH) 2016-07-27 EP disclosed
WO-2010036551-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-04-01 WO disclosed