SCHEMBL7928573

SCHEMBL7928573

COCCN1CCc2cc(NC(=O)c3ccccc3-c3ccc(C(F)(F)F)cc3)ccc2C1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTTP P55157 13/20 0.59
APOB P04114 10/20 0.59
GAA P10253 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
SMO Q99835 1/20 0.50
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8201182 0.95 MTTP (0.57) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL8586390 0.93 MTTP (0.56) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL691193 0.93 MTTP (0.54) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL8208591 0.93 MTTP (0.56) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL8213416 0.91 MTTP (0.58) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL8213404 0.91 MTTP (0.58) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL8200791 0.91 MTTP (0.53) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL8208329 0.90 MTTP (0.57) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL8199851 0.90 MTTP (0.55) MTTPAPOBGAASMN1; SMN2SMO
SCHEMBL692958 0.90 APOB (0.60) MTTPAPOBGAASMN1; SMN2SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099442-A2 Methods of administering apo B-secretion/MTP inhibitors Pfizer Products Inc. (US) 2001-05-16 EP claimed
US-6121283-A Apo B-secretion/MTP inhibitory amides PFIZER INC (US) 2000-09-19 US claimed
EP-0944602-A1 APO B-SECRETION/MTP INHIBITORY AMIDES PFIZER INC. (US) 1999-09-29 EP claimed
WO-1998023593-A1 APO B-SECRETION/MTP INHIBITORY AMIDES PFIZER INC. (US) 1998-06-04 WO claimed
EP-1099442-A2 Methods of administering apo B-secretion/MTP inhibitors Pfizer Products Inc. (US) 2001-05-16 EP disclosed
US-6121283-A Apo B-secretion/MTP inhibitory amides PFIZER INC (US) 2000-09-19 US disclosed
EP-0944602-A1 APO B-SECRETION/MTP INHIBITORY AMIDES PFIZER INC. (US) 1999-09-29 EP disclosed
WO-1998023593-A1 APO B-SECRETION/MTP INHIBITORY AMIDES PFIZER INC. (US) 1998-06-04 WO disclosed