SCHEMBL7928751

SCHEMBL7928751

NS(=O)(=O)c1ccccc1-n1nc(C(F)F)cc1-c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.66
PTGS1 P23219 10/20 0.66
ABCB11 O95342 1/20 0.43
ALDH1A1 P00352 1/20 0.43
PDPK1 O15530 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637047 0.97 PTGS2 (0.63) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL8165901 0.93 PTGS2 (0.62) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL8525009 0.90 PTGS2 (0.65) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL7773921 0.90 PTGS2 (0.65) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL7055102 0.90 PTGS2 (0.64) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8639180 0.88 PTGS2 (0.53) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL8635925 0.88 PTGS2 (0.58) PTGS2PTGS1ABCB11ALDH1A1
Benzenesulfonamide SCHEMBL7927737 0.88 PTGS2 (0.68) PTGS2PTGS1ABCB11ALDH1A1PDPK1
Benzenesulfonamide SCHEMBL8625195 0.88 PTGS2 (0.68) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL8693648 0.87 PTGS2 (0.67) PTGS2PTGS1ABCB11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001527542-A 2001-12-25 JP claimed
EP-0979077-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. Searle & Co. (US) 2000-02-16 EP claimed
WO-1998047509-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1998-10-29 WO claimed
WO-1998016227-A9 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE TREATMENT AND PREVENTION OF NEOPLASIA 1998-07-30 WO claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed