SCHEMBL7932864

SCHEMBL7932864

CCOC(=O)c1sc(C(=O)O)c(-c2ccc(F)cc2)c1-c1ccc(S(=O)(=O)CC)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.49
ALDH1A1 P00352 4/20 0.48
LMNA P02545 2/20 0.48
MAPT P10636 5/20 0.48
KDM4E B2RXH2 3/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TRPM8 Q7Z2W7 1/20 0.48
NPSR1 Q6W5P4 2/20 0.45
PKM P14618 1/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
THRB P10828 1/20 0.43
GRM6 O15303 1/20 0.43
GPR55 Q9Y2T6 1/20 0.43
MAPK14 Q16539 1/20 0.42
CHRNA7 P36544 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6050699 0.91 PTGS2 (0.60) PTGS2ALDH1A1LMNAMAPTKDM4E
SCHEMBL6050619 0.91 PTGS2 (0.60) PTGS2ALDH1A1LMNAMAPTKDM4E
SCHEMBL7162856 0.84 PTGS2 (0.51) PTGS2ALDH1A1MAPTKDM4ENPC1
SCHEMBL6050727 0.82 KDM4E (0.49) PTGS2ALDH1A1LMNAMAPTKDM4E
SCHEMBL6050754 0.82 KDM4E (0.49) PTGS2ALDH1A1LMNAMAPTKDM4E
SCHEMBL6050705 0.77 PTGS2 (0.52) PTGS2KDM4EHPGD
SCHEMBL6050740 0.77 PTGS2 (0.61) PTGS2KDM4EHPGD
SCHEMBL20015818 0.77 MAPT (0.59) PTGS2ALDH1A1LMNAMAPTKDM4E
SCHEMBL12483144 0.75 CHRNA7 (0.60) PTGS2ALDH1A1LMNAMAPTKDM4E
SCHEMBL20015932 0.75 BCL2L1 (0.52) PTGS2ALDH1A1MAPTKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3137648-B2 2001-02-26 JP claimed
EP-0679157-A1 NOVEL 3,4-DIARYL THIOPHENES AND ANALOGS THEREOF HAVING USE AS ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1995-11-02 EP claimed
WO-1994015932-A1 NOVEL 3,4-DIARYL THIOPHENES AND ANALOGS THEREOF HAVING USE AS ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1994-07-21 WO claimed