SCHEMBL7934795

SCHEMBL7934795

Nc1ccccc1NC(=O)/C=C/C=C/C(=O)Nc1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.58
NAMPT P43490 1/20 0.58
ALDH1A1 P00352 5/20 0.58
KDM4E B2RXH2 3/20 0.58
RAB9A P51151 9/20 0.58
NPC1 O15118 8/20 0.58
HDAC2 Q92769 3/20 0.56
HDAC3 O15379 2/20 0.56
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54
SMN1; SMN2 Q16637 4/20 0.53
HDAC4 P56524 2/20 0.53
MEF2D Q14814 1/20 0.53
TP53 P04637 2/20 0.52
EPHA2 P29317 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3263544 0.82 ALDH1A1 (0.66) ALDH1A1KDM4ERAB9ANPC1LMNA
SCHEMBL3263543 0.82 ALDH1A1 (0.66) ALDH1A1KDM4ERAB9ANPC1LMNA
SCHEMBL3228556 0.80 ALDH1A1 (0.82) NAMPTALDH1A1KDM4ERAB9ANPC1
SCHEMBL3228566 0.80 ALDH1A1 (0.82) NAMPTALDH1A1KDM4ERAB9ANPC1
SCHEMBL25722340 0.80 HDAC1 (0.77) HDAC1NAMPTKDM4ERAB9ANPC1
SCHEMBL21232419 0.80 HDAC4 (0.72) HDAC1NAMPTRAB9ANPC1HDAC2
SCHEMBL16016614 0.75 HDAC4 (0.73) HDAC1HDAC2HDAC3LMNAHDAC4
SCHEMBL28410554 0.74 HDAC1 (1.00) HDAC1NAMPTRAB9ANPC1HDAC2
SCHEMBL17667093 0.74 ALDH1A1 (1.00) NAMPTALDH1A1KDM4ERAB9ANPC1
SCHEMBL14164232 0.74 ALDH1A1 (0.71) ALDH1A1KDM4ERAB9ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed