SCHEMBL7936111

SCHEMBL7936111

CCCOc1cc(-c2ccc(C(F)(F)F)cc2)ccc1C=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.46
CYP1A1 P04798 2/20 0.45
CYP1B1 Q16678 2/20 0.45
PSEN1 P49768 2/20 0.43
ALOX5 P09917 2/20 0.43
PPARD Q03181 2/20 0.40
KIF11 P52732 2/20 0.40
ALDH1A1 P00352 4/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTPN1 P18031 1/20 0.38
PTGES O14684 1/20 0.38
PPARG P37231 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MCHR1 Q99705 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL955509 0.89 CYP1A1 (0.46) ERN1CYP1A1CYP1B1PPARDALDH1A1
SCHEMBL23226778 0.86 PSEN1 (0.39) PSEN1ALOX5PPARDKIF11ALDH1A1
SCHEMBL23226562 0.85 MAOB (0.40) PSEN1ALOX5KIF11ALDH1A1MAPT
SCHEMBL23226619 0.85 PSEN1 (0.40) PSEN1ALOX5PPARDKIF11ALDH1A1
SCHEMBL23226546 0.85 CACNA1B (0.41) PSEN1ALOX5KIF11KDM4EMCHR1
SCHEMBL953869 0.82 PTGDR2 (0.48) CYP1A1CYP1B1PSEN1ALOX5PPARD
SCHEMBL7943031 0.78 ERN1 (0.49) ERN1ALDH1A1MAPTHPGDHTT
SCHEMBL957465 0.77 CYP2C19 (0.50) CYP1A1CYP1B1ALDH1A1MAPTHPGD
SCHEMBL23226899 0.77 EPHX2 (0.53) KDM4E
SCHEMBL7946267 0.77 PPARD (0.41) CYP1A1CYP1B1PSEN1ALOX5PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015653-A1 PYRIMIDINE DERIVATIVES AS ACTIVATORS OF SOLUBLE GUANYLATE CYCLASE SMITHKLINE BEECHAM CORPORATION (US) 2010-02-11 WO disclosed
WO-2009071504-A1 2,6-DISUBSTITUTED PYRIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-11 WO disclosed