SCHEMBL7946267

SCHEMBL7946267

CCCOc1cc(-c2ccc(C(F)(F)F)cc2)ccc1CBr

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 6/20 0.41
KIF11 P52732 4/20 0.38
TRPV1 Q8NER1 1/20 0.38
MCHR1 Q99705 2/20 0.38
ALOX5 P09917 1/20 0.37
PSEN1 P49768 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
AGXT P21549 1/20 0.37
SCN8A Q9UQD0 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
CYP1A1 P04798 2/20 0.36
CYP1B1 Q16678 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7935451 0.86 PPARD (0.43) PPARDKIF11TRPV1MCHR1ALOX5
SCHEMBL7944912 0.78 TSHR (0.39)
SCHEMBL7936111 0.77 ERN1 (0.46) PPARDKIF11MCHR1ALOX5PSEN1
SCHEMBL4602156 0.76 PTPN11 (0.60) PPARDALOX5PSEN1PPARA
SCHEMBL3230214 0.74 RXRA (0.50) KIF11PSEN1AGXT
SCHEMBL2056314 0.74 CYP1A1 (0.56) PPARDKIF11PPARACYP1A1CYP1B1
SCHEMBL3235607 0.72 HPGD (0.50)
SCHEMBL14610858 0.72 PTPN11 (0.46) PPARDKIF11MCHR1ALOX5PSEN1
SCHEMBL12650491 0.72 KIF11 (0.55) PPARDKIF11MCHR1PPARGPPARA
SCHEMBL13756268 0.71 KIF11 (0.40) PPARDKIF11MCHR1ALOX5PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015653-A1 PYRIMIDINE DERIVATIVES AS ACTIVATORS OF SOLUBLE GUANYLATE CYCLASE SMITHKLINE BEECHAM CORPORATION (US) 2010-02-11 WO disclosed
WO-2009071504-A1 2,6-DISUBSTITUTED PYRIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-11 WO disclosed