SCHEMBL7937713

SCHEMBL7937713

Nc1cccc(OC(F)(F)F)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MPL P40238 1/20 0.40
GRIA1 P42261 5/20 0.36
CACNG8 Q8WXS5 5/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
P2RX7 Q99572 3/20 0.35
GRIN2B Q13224 1/20 0.35
ALDH1A1 P00352 2/20 0.34
ADRA2B P18089 1/20 0.34
PTGS1 P23219 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 3/20 0.34
MAPT P10636 2/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
NR4A2 P43354 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14744548 0.84 MPL (0.41) MPLALDH1A1KDM4EMAPTL3MBTL1
SCHEMBL8074941 0.82 PDE2A (0.33) MPLGRIN2BALDH1A1TDP1MAPT
SCHEMBL3790638 0.82 KCNH2 (0.45) CYP1A2CYP3A4CYP2C19ALDH1A1ADRA2B
SCHEMBL2848722 0.79 MPL (0.41) MPLCYP3A4ALDH1A1ADRA2BPTGS1
SCHEMBL8653715 0.79 GRIA1 (0.48) GRIA1CACNG8CYP1A2CYP3A4CYP2C19
SCHEMBL29893374 0.79 ALDH1A1 (0.50) MPLCYP1A2CYP3A4CYP2C19GRIN2B
SCHEMBL112134 0.79 ALDH1A1 (0.50) MPLCYP1A2CYP3A4CYP2C19GRIN2B
SCHEMBL12480337 0.78 MPL (0.51) MPLCYP3A4ALDH1A1ADRA2BPTGS1
Hydrochloric Acid SCHEMBL4379610 0.77 ALDH1A1 (0.48) MPLCYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL21603543 0.76 GRIA1 (0.42) MPLGRIA1CACNG8P2RX7GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235939-B1 TRIFLUOROALKOXY-5-CHLOROANILINE BAYER AKTIENGESELLSCHAFT (DE) 2001-05-22 US claimed
EP-0546391-A2 Process for the preparation of fluorine containing anilines. BAYER AG (DE) 1993-06-16 EP claimed
US-6235939-B1 TRIFLUOROALKOXY-5-CHLOROANILINE BAYER AKTIENGESELLSCHAFT (DE) 2001-05-22 US disclosed
US-6077973-A Process for the preparation of anilines which contain fluorine and new anilines which contain fluorine BAYER AKTIENGESELLSCHAFT (DE) 2000-06-20 US disclosed
EP-0546391-B1 Process for the preparation of fluorine containing anilines. BAYER AG (DE) 1996-05-08 EP disclosed
EP-0546391-A2 Process for the preparation of fluorine containing anilines. BAYER AG (DE) 1993-06-16 EP disclosed