SCHEMBL7938628

SCHEMBL7938628

COC(=O)c1ccc(-c2coc(-c3cncc(I)c3)n2)cn1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.42
MAPK1 P28482 1/20 0.40
HPGD P15428 1/20 0.38
ALOX5AP P20292 1/20 0.38
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
S1PR1 P21453 1/20 0.35
ENPP3 O14638 1/20 0.35
ENPP1 P22413 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
LCK P06239 1/20 0.34
SMO Q99835 2/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
NOTUM Q6P988 1/20 0.34
PDE10A Q9Y233 1/20 0.34
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1001318 0.88 DYRK1A (0.43) DYRK1AMAPK1HPGDALOX5APHDAC1
SCHEMBL1002385 0.76 GRM5 (0.47) DYRK1AMAPK1HPGDALOX5APENPP3
SCHEMBL1002632 0.74 ABL1 (0.41) DYRK1AMAPK1HPGDALOX5AP
SCHEMBL1004185 0.71 MAPK1 (0.44) DYRK1AMAPK1HPGDALOX5APS1PR1
SCHEMBL27237310 0.70 HDAC1 (0.55) HDAC1HDAC8HDAC6
SCHEMBL1002350 0.69 HDAC1 (0.48) HPGDHDAC1HDAC8HDAC6
SCHEMBL1002558 0.69 MAPK1 (0.43) DYRK1AMAPK1HPGDALOX5APPDE10A
SCHEMBL24370250 0.68 MAPK1 (0.50) DYRK1AMAPK1HPGDCYP11B1CYP11B2
SCHEMBL1004945 0.67 ALDH1A1 (0.40) DYRK1AMAPK1HPGDALOX5APS1PR1
SCHEMBL5845581 0.67 MAPK1 (0.65) DYRK1AMAPK1HPGDLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010017079-A1 OXAZOLE DERIVATIVES USEFUL AS INHIBITORS OF FAAH MERCK & CO., INC. (US) 2010-02-11 WO disclosed