SCHEMBL7939207

SCHEMBL7939207

C=C(O)c1c(F)cccc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RORC P51449 9/20 0.42
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
HSD11B1 P28845 1/20 0.37
CYP2C9 P11712 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C19 P33261 2/20 0.37
PTGS2 P35354 1/20 0.37
TXNRD1 Q16881 1/20 0.37
ITGA4 P13612 2/20 0.36
ITGB1 P05556 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
RORB Q92753 1/20 0.36
STIM1 Q13586 1/20 0.35
ORAI1 Q96D31 1/20 0.35
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14534757 0.82 CES2 (0.39) RORCCES2CES1HSD11B1PTGS2
SCHEMBL503596 0.80 CES2 (0.50) RORCCES2CES1CYP2C9CYP3A4
SCHEMBL21518072 0.78 CES2 (0.48) RORCCES2CES1CYP2C9CYP3A4
SCHEMBL17054742 0.74 CES2 (0.39) RORCCES2CES1ITGA4RORB
SCHEMBL476764 0.74 CES2 (0.48) RORCCES2CES1CYP2C9CYP3A4
SCHEMBL716995 0.74 CES2 (0.48) RORCCES2CES1PTGS2MEN1
SCHEMBL30313345 0.74 CES2 (0.48) RORCCES2CES1PTGS2MEN1
SCHEMBL20560651 0.74 CES2 (0.39) RORCCES2CES1CYP2C9CYP3A4
SCHEMBL3708513 0.74 CES2 (0.48) RORCCES2CES1PTGS2ITGA4
Hydrochloric Acid SCHEMBL4371024 0.73 CES2 (0.47) RORCCES2CES1PTGS2ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020548-A1 GLYT1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-02-25 WO disclosed