SCHEMBL7941737

SCHEMBL7941737

CC(C)(C)OC(=O)CN(CC(=O)OC(C)(C)C)C(CO)CCCCCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 4/20 0.46
KCNH2 Q12809 5/20 0.41
TSHR P16473 1/20 0.39
NR1H3 Q13133 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
EPHX1 P07099 1/20 0.36
PTGES O14684 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3132273 0.96 NR1D1 (0.48) NR1D1KCNH2TSHRNR1H3PPARG
SCHEMBL13014392 0.91 NR1D1 (0.49) NR1D1KCNH2TSHRNR1H3PPARG
SCHEMBL15388528 0.83 NR1D1 (0.48) NR1D1KCNH2TSHRNR1H3PPARG
SCHEMBL17986044 0.81 NR1D1 (0.42) NR1D1KCNH2MMP1MMP2MMP9
SCHEMBL3773796 0.80 NR1D1 (0.42) NR1D1KCNH2MAPTL3MBTL1
SCHEMBL17986065 0.77 NR1D1 (0.43) NR1D1KCNH2
SCHEMBL3773804 0.77 NR1D1 (0.40) NR1D1KCNH2MAPTL3MBTL1
SCHEMBL13014059 0.76 NR1D1 (0.39) NR1D1KCNH2MAPTL3MBTL1
SCHEMBL13014102 0.76 NR1D1 (0.52) NR1D1KCNH2TSHRNR1H3PPARG
SCHEMBL15388422 0.76 NR1D1 (0.52) NR1D1KCNH2TSHRNR1H3PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010011367-A2 BIMODAL LIGANDS WITH MACROCYCLIC AND ACYCLIC BINDING MOIETIES, COMPLEXES AND COMPOSITIONS THEREOF, AND METHODS OF USING ILLINOIS INSTITUTE OF TECHNOLOGY (US) 2010-01-28 WO disclosed