SCHEMBL794302

SCHEMBL794302

Cc1ccncc1N1CCc2sc3ccc(F)cc3c2C1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 8/20 0.58
CYP3A4 P08684 6/20 0.58
CYP1A2 P05177 2/20 0.36
MAPT P10636 1/20 0.35
TDO2 P48775 1/20 0.35
HRH4 Q9H3N8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL798823 0.79 CYP17A1 (0.52) CYP17A1CYP3A4MAPTTDO2HRH4
SCHEMBL15465685 0.75 CYP17A1 (0.52) CYP17A1CYP3A4HRH4
SCHEMBL3782220 0.71 CYP17A1 (0.52) CYP17A1CYP3A4
SCHEMBL29412530 0.66 KCNQ2 (0.47) CYP17A1CYP3A4
SCHEMBL807981 0.65 CYP17A1 (0.39) CYP17A1CYP3A4
SCHEMBL18949756 0.65 MAPT (0.54) CYP3A4CYP1A2MAPT
SCHEMBL793782 0.65 CDC7 (0.40) CYP17A1CYP3A4
SCHEMBL793474 0.65 CYP11B2 (0.41) CYP17A1CYP1A2MAPT
SCHEMBL794339 0.65 CYP17A1 (0.37) CYP17A1CYP3A4CYP1A2MAPT
SCHEMBL793824 0.63 CYP11B2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627648-A1 17aHYDROXYLASE/C17,20-LYASE INHIBITORS Novartis AG (CH) 2013-08-21 EP disclosed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO disclosed