SCHEMBL7943767

SCHEMBL7943767

COc1ccc2c(c1)/C(=C/C#N)CCCC2

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.47
CYP11B2 P19099 6/20 0.47
ABCB1 P08183 1/20 0.44
MAOB P27338 2/20 0.42
NQO2 P16083 2/20 0.41
MTNR1A P48039 2/20 0.41
MTNR1B P49286 2/20 0.41
ALDH1A1 P00352 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP11B1 P15538 2/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAOA P21397 1/20 0.39
NPY5R Q15761 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7943769 1.00 CYP19A1 (0.47) CYP19A1CYP11B2ABCB1MAOBNQO2
SCHEMBL7951341 0.97 CYP19A1 (0.47) CYP19A1CYP11B2ABCB1MAOBNQO2
SCHEMBL7951337 0.97 CYP19A1 (0.47) CYP19A1CYP11B2ABCB1MAOBNQO2
SCHEMBL1688133 0.97 CYP19A1 (0.47) CYP19A1CYP11B2ABCB1MAOBNQO2
SCHEMBL4688568 0.91 CYP19A1 (0.56) CYP19A1CYP11B2MAOBNQO2MTNR1A
SCHEMBL4688774 0.91 CYP19A1 (0.56) CYP19A1CYP11B2MAOBNQO2MTNR1A
SCHEMBL31028072 0.91 CYP19A1 (0.56) CYP19A1CYP11B2MAOBNQO2MTNR1A
SCHEMBL4688567 0.91 CYP19A1 (0.56) CYP19A1CYP11B2MAOBNQO2MTNR1A
SCHEMBL7952133 0.85 ADCY8 (0.36) CYP19A1CYP11B2ABCB1MAOBNQO2
SCHEMBL7952131 0.85 ADCY8 (0.36) CYP19A1CYP11B2ABCB1MAOBNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235789-B1 GLANDULAR DISORDERS; SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0781271-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-07-02 EP disclosed
WO-1996008466-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-21 WO disclosed