SCHEMBL7944113

SCHEMBL7944113

CN(C)c1cccc(N)c1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.47
NEK2 P51955 1/20 0.47
LIMK1 P53667 1/20 0.47
DYRK1A Q13627 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
GAA P10253 6/20 0.43
MAPT P10636 6/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 6/20 0.40
TSHR P16473 4/20 0.40
CYP3A4 P08684 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PIK3CA P42336 1/20 0.39
MCL1 Q07820 1/20 0.37
KMT2A Q03164 2/20 0.36
CA2 P00918 1/20 0.36
CD44 P16070 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9614284 0.76 CHEK1 (0.50) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL9566860 0.76 MAPT (0.46) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL29707613 0.75 CHEK1 (0.60) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL113870 0.75 CHEK1 (0.60) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL29922382 0.74 CHEK1 (0.79) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL2886998 0.74 CHEK1 (0.79) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL31689542 0.74 CHEK1 (0.79) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL2886968 0.74 CYP3A4 (0.59) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL2015386 0.74
Hydrochloric Acid SCHEMBL6378551 0.73 CHEK1 (0.58) CHEK1NEK2LIMK1DYRK1ACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6307087-B1 USE OF CATALYSTS COMPRISING THESE LIGANDS IN TRANSITION METAL-CATALYZED CARBON-HETEROATOM AND CARBON-CARBON BOND-FORMING REACTIONS. MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2001-10-23 US disclosed