SCHEMBL794501

SCHEMBL794501

CCOC(=O)C1Cc2ccc(Br)cc2C1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.49
ALDH1A1 P00352 7/20 0.49
KDM4E B2RXH2 5/20 0.49
MEN1 O00255 6/20 0.47
MAPK1 P28482 4/20 0.47
TSHR P16473 3/20 0.45
ADRA2A P08913 1/20 0.44
PNMT P11086 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
TDP2 O95551 1/20 0.44
GAA P10253 2/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
POLB P06746 2/20 0.42
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CCR5 P51681 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31537552 1.00 KMT2A (0.49) KMT2AALDH1A1KDM4EMEN1MAPK1
SCHEMBL10529754 0.89 MAPK1 (0.46) KMT2AALDH1A1KDM4EMEN1MAPK1
SCHEMBL30437653 0.89 MAPK1 (0.46) KMT2AALDH1A1KDM4EMEN1MAPK1
SCHEMBL30437369 0.83 KMT2A (0.47) KMT2AALDH1A1ADRA2APNMTADRA2B
SCHEMBL1339915 0.83 KMT2A (0.47) KMT2AALDH1A1ADRA2APNMTADRA2B
SCHEMBL15823733 0.82 KDM4E (0.49) KMT2AALDH1A1KDM4EMEN1GAA
SCHEMBL22070557 0.81 TP53 (0.45) KMT2AALDH1A1KDM4EMEN1MAPK1
SCHEMBL8569044 0.81 KMT2A (0.45) KMT2AALDH1A1KDM4EMEN1MAPK1
SCHEMBL8569048 0.81 KMT2A (0.45) KMT2AALDH1A1KDM4EMEN1MAPK1
SCHEMBL8569043 0.81 KMT2A (0.45) KMT2AALDH1A1KDM4EMEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023225162-A1 ANTIVIRAL INDOLINYL COMPOUNDS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2023-11-23 WO disclosed
EP-2735562-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS INC (US) 2023-11-15 EP disclosed
EP-2735562-B2 Estrogen receptor modulators and uses thereof SERAGON PHARMACEUTICALS INC (US) 2023-11-15 EP disclosed
US-20230132370-A9 CRYSTAL FORMS OF THIAZOLE COMPOUND AND APPLICATION THEREOF MEDSHINE DISCOVERY INC. (CN) 2023-04-27 US disclosed
US-20230132370-A9 CRYSTAL FORMS OF THIAZOLE COMPOUND AND APPLICATION THEREOF MEDSHINE DISCOVERY INC. (CN) 2023-04-27 US disclosed
EP-3566749-A1 THIAZOLE DERIVATIVE AND APPLICATIONS THEREOF Medshine Discovery Inc. (CN) 2019-11-13 EP disclosed
US-9868704-B2 Estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2018-01-16 US disclosed
US-9868704-B2 Estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2018-01-16 US disclosed
US-9868704-B2 Estrogen receptor modulators and uses thereof GENENTECH, INC. (US) 2018-01-16 US disclosed
EP-2934533-B1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME (US) 2017-11-15 EP disclosed
US-20130231333-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-09-05 US disclosed
US-20130231333-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2013-09-05 US disclosed
EP-2616445-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF Aragon Pharmaceuticals, Inc. (US) 2013-07-24 EP disclosed
WO-2013062892-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2013-05-02 WO disclosed
WO-2012037411-A9 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed
WO-2012037411-A2 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ARAGON PHARMACEUTICALS, INC. (US) 2012-03-22 WO disclosed
EP-0135177-B1 BENZOCYCLOALKANE DERIVATIVES DAIICHI SEIYAKU CO., LTD. (JP) 1989-12-06 EP disclosed
US-4777257-A CARDIOVASCULAR DISORDERS DAIICHI SEIYAKU CO., LTD. (JP) 1988-10-11 US disclosed
US-4665188-A Certain [(1-imidazolyl)-lower-alkylene]-tetrahydronaphthalenecarboxylic acids or corresponding idan-carboxylic acids which are thromboxane A2 DAIICHI SEIYAKU CO., LTD. (JP) 1987-05-12 US disclosed
EP-0135177-A2 Benzocycloalkane derivatives DAIICHI SEIYAKU CO., LTD. (JP) 1985-03-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230132370-A9 CRYSTAL FORMS OF THIAZOLE COMPOUND AND APPLICATION THEREOF ZC3HAV1L, ZC3HAV1, RPL35 KMT2A 3913/4885ALDH1A1 1605/4885KDM4E 3127/4885
US-20130231333-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF ESR2, ESRRG, GPER1 KMT2A 2760/4885ALDH1A1 1138/4885KDM4E 2775/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.