SCHEMBL7945448

SCHEMBL7945448

CCc1ccc(-c2coc(-c3ccc(F)cc3)n2)cn1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
KDM5B Q9UGL1 1/20 0.42
LMNA P02545 1/20 0.41
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
HPGD P15428 1/20 0.39
ENPP3 O14638 3/20 0.39
ENPP1 P22413 3/20 0.39
PDE4B Q07343 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27903340 0.85 HDAC1 (0.41) MMP13HDAC1HDAC8HDAC6KDM5B
SCHEMBL1002924 0.83 LMNA (0.39) MMP13HDAC1HDAC8HDAC6KDM5B
SCHEMBL14294336 0.79 LMNA (0.52) HDAC1HDAC8HDAC6LMNAKMT2A
SCHEMBL1001407 0.78 HDAC1 (0.42) MMP13HDAC1HDAC8HDAC6KDM5B
SCHEMBL1002194 0.77 KDM5B (0.41) MMP13HDAC1HDAC8HDAC6KDM5B
SCHEMBL15802660 0.77 KDM4E (0.42) MMP13HDAC1HDAC8HDAC6KDM5B
SCHEMBL1002193 0.77 KDM5B (0.41) MMP13HDAC1HDAC8HDAC6KDM5B
SCHEMBL1004600 0.77 KDM5B (0.41) MMP13HDAC1HDAC8HDAC6KDM5B
SCHEMBL1002137 0.77 KDM5B (0.41) MMP13HDAC1HDAC8HDAC6KDM5B
SCHEMBL15520374 0.77 KDM5B (0.41) MMP13HDAC1HDAC8HDAC6KDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010017079-A1 OXAZOLE DERIVATIVES USEFUL AS INHIBITORS OF FAAH MERCK & CO., INC. (US) 2010-02-11 WO disclosed