SCHEMBL7946639

SCHEMBL7946639

Cc1c(-c2nc3c(F)c(F)cc(F)c3s2)c2cc(Cl)ccc2n1CC(=O)O.Cc1c(-c2nc3c(F)c(F)cc(F)c3s2)c2ccc(Cl)cc2n1CC(=O)O.Cc1ccc2c(c1)c(-c1nc3c(F)c(F)cc(F)c3s1)c(C)n2CC(=O)O.Cc1cccc2c(-c3nc4c(F)c(F)cc(F)c4s3)c(C)n(CC(=O)O)c12.Cc1cccc2c1c(-c1nc3c(F)c(F)cc(F)c3s1)c(C)n2CC(=O)O

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 10/20 0.48
AKR1A1 P14550 9/20 0.48
PTGDR2 Q9Y5Y4 11/20 0.43
PTGS1 P23219 2/20 0.43
CYP2C9 P11712 1/20 0.43
SLC6A4 P31645 1/20 0.43
CYP2C19 P33261 1/20 0.43
PTGS2 P35354 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6140102 0.84 AKR1B1 (0.56) AKR1B1AKR1A1PTGDR2PTGS1
SCHEMBL7755666 0.83 AKR1B1 (0.58) AKR1B1AKR1A1PTGDR2PTGS1CYP2C9
SCHEMBL7754910 0.83 AKR1B1 (0.58) AKR1B1AKR1A1PTGDR2PTGS1CYP2C9
SCHEMBL7755683 0.83 AKR1A1 (0.58) AKR1B1AKR1A1PTGDR2PTGS1
SCHEMBL7751532 0.81 AKR1B1 (0.58) AKR1B1AKR1A1PTGDR2PTGS1CYP2C9
SCHEMBL7951912 0.81 AKR1A1 (0.60) AKR1B1AKR1A1PTGDR2PTGS1CYP2C9
SCHEMBL2098715 0.80 AKR1B1 (0.70) AKR1B1AKR1A1PTGDR2
Water SCHEMBL5501664 0.79 AKR1B1 (0.69) AKR1B1AKR1A1PTGDR2
SCHEMBL2820038 0.79 AKR1B1 (0.56) AKR1B1AKR1A1PTGDR2
SCHEMBL5888935 0.79 AKR1B1 (0.56) AKR1B1AKR1A1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001064205-A2 COMPOSITIONS CONTAINING A SUBSTITUTED INDOLEALKANOIC ACID AND AN ANGIOTENSIN CONVERTING ENZYME INHIBITOR THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2001-09-07 WO disclosed