SCHEMBL7946732

SCHEMBL7946732

CC#CCNc1cnc(C(=O)Nc2ccc(F)c(CNc3cccnc3N)c2)cn1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 14/20 0.57
HDAC3 O15379 2/20 0.44
NCOR1 O75376 2/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
BACE2 Q9Y5Z0 1/20 0.42
TMEM97 Q5BJF2 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
AURKA O14965 1/20 0.39
AURKB Q96GD4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12303597 0.90 BACE1 (0.54) BACE1HDAC3NCOR1HDAC1HDAC2
SCHEMBL7942878 0.87 BACE1 (0.75) BACE1BACE2
SCHEMBL7939911 0.85 BACE1 (0.64) BACE1BACE2
SCHEMBL7940775 0.85 BACE1 (0.59) BACE1HDAC3NCOR1HDAC1HDAC2
SCHEMBL7933179 0.85 BACE1 (0.76) BACE1HDAC3NCOR1HDAC1HDAC2
SCHEMBL7941880 0.85 SMN1; SMN2 (0.57) BACE1BACE2NPC1RAB9ASMN1; SMN2
SCHEMBL7941874 0.84 BACE1 (0.60) BACE1BACE2AURKAAURKB
SCHEMBL7944835 0.84 BACE1 (0.54) BACE1HDAC3NCOR1HDAC1HDAC2
SCHEMBL7941875 0.83 BACE1 (0.73) BACE1BACE2
SCHEMBL7945376 0.83 BACE1 (0.54) BACE1BACE2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010047372-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY 塩野義製薬株式会社 (JP) 2010-04-29 WO disclosed