SCHEMBL7947489

SCHEMBL7947489

Cc1ccc(-c2cc(C(=O)N[C@@H](Cl)CO)cc(-c3cccc(F)c3F)c2)nc1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 11/20 0.50
P2RX2 Q9UBL9 10/20 0.50
NR1I2 O75469 3/20 0.50
CTSA P10619 2/20 0.43
CYP2C9 P11712 2/20 0.41
UGT1A1 P22309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171499 0.90 P2RX3 (0.61) P2RX3P2RX2NR1I2
SCHEMBL2171032 0.85 P2RX3 (0.49) P2RX3P2RX2NR1I2CTSACYP2C9
SCHEMBL2187309 0.82 P2RX3 (0.56) P2RX3P2RX2NR1I2CTSACYP2C9
SCHEMBL2172363 0.82 P2RX3 (0.49) P2RX3P2RX2NR1I2CTSACYP2C9
SCHEMBL2172956 0.81 NR1I2 (0.45) P2RX3P2RX2NR1I2CTSA
SCHEMBL2170986 0.80 NR1I2 (0.45) P2RX3P2RX2NR1I2CTSA
SCHEMBL2171462 0.79 P2RX3 (0.53) P2RX3P2RX2NR1I2
SCHEMBL2171457 0.79 P2RX3 (0.53) P2RX3P2RX2NR1I2
SCHEMBL2174361 0.78 P2RX3 (0.48) P2RX3P2RX2NR1I2
SCHEMBL2171711 0.75 CYP3A4 (0.46) P2RX3P2RX2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010033168-A2 AMIDE COMPOUNDS, COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2010-03-25 WO disclosed