SCHEMBL7948387

SCHEMBL7948387

O=C(O)COc1cccc2c1ccn2CCOCCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.55
PPARG P37231 3/20 0.49
PPARA Q07869 3/20 0.49
HTR6 P50406 1/20 0.46
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
BAD Q92934 1/20 0.44
BCL2 P10415 1/20 0.43
HRH2 P25021 2/20 0.42
PLA2G2A P14555 2/20 0.42
ROCK1 Q13464 1/20 0.41
RAB9A P51151 1/20 0.41
PTPN7 P35236 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958296 0.93 MCL1 (0.56) MCL1PPARGPPARAHTR6KDM4E
SCHEMBL7959220 0.85 MCL1 (0.59) MCL1PPARGPPARAHTR6KDM4E
SCHEMBL7960467 0.84 MCL1 (0.53) MCL1PPARGPPARAHTR6KDM4E
SCHEMBL7958447 0.83 MCL1 (0.54) MCL1PPARGPPARAHTR6KDM4E
SCHEMBL7959506 0.80 MCL1 (0.60) MCL1PPARGPPARAHTR6KDM4E
SCHEMBL7959081 0.80 MCL1 (0.53) MCL1PPARGPPARAHTR6KDM4E
SCHEMBL7948724 0.80 MCL1 (0.55) MCL1PPARGPPARAHTR6KDM4E
SCHEMBL7960155 0.79 MCL1 (0.59) MCL1PPARGPPARAHTR6KDM4E
SCHEMBL7958387 0.79 HTR2C (0.51) MCL1HTR6KDM4EALDH1A1BAD
SCHEMBL7962451 0.79 HTR6 (0.47) MCL1HTR6TDP1BADBCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6323235-B1 CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS AND ENZYME INHIBITORS OHTAKE ATSUSHI (JP) 2001-11-27 US disclosed
US-6043264-A A THROMBOXANE A2 RECEPTOR ANTAGONIST FOR TREATING HYPERTENSION, THROMBOSIS, ISCHEMIC HEART DISEASES, CIRCULATORY DISEASES, ARTERIOSCLEROSIS, PLATELET FUNCTION DISORDER, HYPERLIPIDEMIA, NEPHRITIS OR ASTHMA TORAY INDUSTRIES, INC. (JP) 2000-03-28 US disclosed
EP-0751126-A1 BENZENE-FUSED HETEROCYCLIC DERIVATIVE AND USE OF THE SAME TORAY INDUSTRIES, INC. (JP) 1997-01-02 EP disclosed