SCHEMBL7948769

SCHEMBL7948769

C=Cc1ccc2c(ccc(=O)n2C)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRPF1 P55201 16/20 0.57
BRD4 O60885 5/20 0.50
BRD9 Q9H8M2 5/20 0.50
CA12 O43570 1/20 0.50
CA9 Q16790 1/20 0.50
KAT2B Q92831 1/20 0.50
BRD1 O95696 9/20 0.43
BRPF3 Q9ULD4 4/20 0.43
CYP2A6 P11509 1/20 0.41
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
BCL6 P41182 1/20 0.36
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1771879 0.77 BRPF1 (0.62) BRPF1BRD4BRD9CA12CA9
SCHEMBL18000169 0.75 MEN1 (0.42)
SCHEMBL422084 0.74 BRPF1 (0.65) BRPF1BRD4BRD9CA12CA9
SCHEMBL8556776 0.73 BRPF1 (0.62) BRPF1BRD4BRD9CA12CA9
SCHEMBL7085783 0.73 BRPF1 (1.00) BRPF1BRD4BRD9CA12CA9
SCHEMBL2172818 0.73 BRPF1 (0.62) BRPF1BRD4BRD9CA12CA9
SCHEMBL31202712 0.73 BRPF1 (0.62) BRPF1BRD4BRD9CA12CA9
SCHEMBL3147477 0.73 CYP2A6 (0.68) CYP2A6PIK3CB
SCHEMBL9257087 0.73 BRPF1 (0.62) BRPF1BRD4BRD9CA12CA9
SCHEMBL31596823 0.73 CYP2A6 (0.68) CYP2A6PIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010035745-A1 HETEROCYCLIC BIARYL DERIVATIVE, AND PDE INHIBITOR COMPRISING SAME AS ACTIVE INGREDIENT 杏林製薬株式会社 (JP) 2010-04-01 WO disclosed