SCHEMBL7948880

SCHEMBL7948880

Bc1ccc2c(c1)C1(CC(c3ccccc3)O2)N=C(N)N(CC)C1=O

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 14/20 0.44
CTSD P07339 12/20 0.44
BACE2 Q9Y5Z0 1/20 0.41
AKR1B1 P15121 1/20 0.37
CTSE P14091 1/20 0.32
ABCB1 P08183 1/20 0.32
AR P10275 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
LMNA P02545 1/20 0.32
ADORA3 P0DMS8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7960752 0.89 BACE1 (0.41) BACE1CTSDBACE2AKR1B1
SCHEMBL2376968 0.88 BACE1 (0.45) BACE1CTSDBACE2AKR1B1
SCHEMBL7962869 0.88 BACE1 (0.46) BACE1CTSDAKR1B1AR
SCHEMBL7959217 0.87 BACE1 (0.35) BACE1CTSDBACE2AKR1B1ABCB1
SCHEMBL2376546 0.81 BACE1 (0.53) BACE1CTSDBACE2
SCHEMBL12245450 0.81 BACE1 (0.51) BACE1CTSD
SCHEMBL2375775 0.81 BACE1 (0.46) BACE1CTSDBACE2AKR1B1
SCHEMBL2375565 0.81 BACE1 (0.46) BACE1CTSDBACE2AKR1B1
SCHEMBL2376874 0.78 BACE1 (0.42) BACE1CTSDBACE2AKR1B1
SCHEMBL2387038 0.77 BACE1 (0.49) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed