SCHEMBL7962869

SCHEMBL7962869

Bc1ccc2c(c1)C1(CC(c3ccccc3)O2)N=C(N)N(CC(F)(F)F)C1=O

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.46
CTSD P07339 6/20 0.46
AKR1B1 P15121 1/20 0.37
AR P10275 2/20 0.33
SCN9A Q15858 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2375593 0.89 BACE1 (0.46) BACE1CTSDAKR1B1
SCHEMBL7948880 0.88 BACE1 (0.44) BACE1CTSDAKR1B1AR
SCHEMBL7960752 0.87 BACE1 (0.41) BACE1CTSDAKR1B1SCN9A
SCHEMBL2375464 0.82 BACE1 (0.52) BACE1CTSD
SCHEMBL12244930 0.82 BACE1 (0.52) BACE1CTSD
SCHEMBL7959217 0.77 BACE1 (0.35) BACE1CTSDAKR1B1AR
SCHEMBL2376968 0.76 BACE1 (0.45) BACE1CTSDAKR1B1
SCHEMBL2376466 0.76 BACE1 (0.47) BACE1CTSDAKR1B1
SCHEMBL12246268 0.76 BACE1 (0.41) BACE1CTSDAKR1B1
SCHEMBL2376874 0.76 BACE1 (0.42) BACE1CTSDAKR1B1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed