SCHEMBL7950709

SCHEMBL7950709

N#C/N=C1/CC2(CCCN(c3ncccn3)C2)Oc2ccc(-c3cccc(C#N)c3)cc21

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 1/20 0.42
LRRK2 Q5S007 9/20 0.39
BACE1 P56817 2/20 0.37
USP30 Q70CQ3 5/20 0.36
PRKCQ Q04759 2/20 0.35
MAP4K1 Q92918 2/20 0.35
PRKCH P24723 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7959648 0.89 SLC6A7 (0.46) SLC6A7LRRK2BACE1USP30PRKCQ
SCHEMBL7962016 0.88 USP2 (0.37) LRRK2BACE1USP30PRKCQMAP4K1
SCHEMBL7957828 0.88 SLC6A7 (0.45) SLC6A7LRRK2BACE1USP30
SCHEMBL2375582 0.79 BACE1 (0.41) LRRK2BACE1
SCHEMBL2375588 0.79 BACE1 (0.41) LRRK2BACE1
SCHEMBL7964219 0.78 BACE1 (0.38) LRRK2BACE1CYP1A2CYP3A4TP53
SCHEMBL7949771 0.78 BACE1 (0.39) LRRK2BACE1
SCHEMBL12246411 0.78 BACE1 (0.39) LRRK2BACE1
SCHEMBL1820029 0.78 BACE1 (0.45) BACE1
SCHEMBL1820031 0.78 BACE1 (0.45) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921359-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-12-30 US disclosed
EP-2324032-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2014-10-01 EP disclosed
US-8450308-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2013-05-28 US disclosed
US-20110218192-A1 Inhibitors Of Beta-Secretase VITAE PHARMACEUTICALS, INC. (US) 2011-09-08 US disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110218192-A1 Inhibitors Of Beta-Secretase BACE1, BACE2, APP SLC6A7 965/4885LRRK2 401/4885BACE1 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.