SCHEMBL7954729

SCHEMBL7954729

OCCC1(c2ccc(F)cc2F)CCNC1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 14/20 0.42
SLC6A3 Q01959 14/20 0.42
SLC6A4 P31645 13/20 0.42
CYP2D6 P10635 9/20 0.41
KCNH2 Q12809 2/20 0.38
DPP4 P27487 1/20 0.33
BACE1 P56817 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8807923 0.82 SLC6A2 (0.43) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2
SCHEMBL5592232 0.82 SLC6A4 (0.41) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2
SCHEMBL6993490 0.79 SLC6A3 (0.52) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2
SCHEMBL6993234 0.75 SLC6A4 (0.56) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2
Hydrochloric Acid SCHEMBL7000511 0.74 SLC6A4 (0.54) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2
SCHEMBL3108178 0.74 CCNT1 (0.40) SLC6A2SLC6A3SLC6A4DPP4BACE1
SCHEMBL16585059 0.73 BACE1 (0.39) BACE1HDAC3HDAC1HDAC2HDAC6
SCHEMBL30232775 0.72 SLC6A4 (0.46) SLC6A2SLC6A3SLC6A4DPP4BACE1
SCHEMBL30232387 0.72 SLC6A4 (0.46) SLC6A2SLC6A3SLC6A4KCNH2DPP4
SCHEMBL3119870 0.72 BACE1 (0.36) SLC6A2SLC6A3SLC6A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329392-B1 ANTIALLERGENS AVENTIS PHARMACEUTICALS, INC. 2001-12-11 US disclosed
EP-0777666-B1 SUBSTITUTED PIPERIDINES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES MERRELL PHARMA INC (US) 1999-03-03 EP disclosed
EP-0777666-A1 NOVEL SUBSTITUTED PIPERIDINES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES MERRELL PHARMACEUTICALS INC. (US) 1997-06-11 EP disclosed
WO-1996006094-A1 NOVEL SUBSTITUTED PIPERIDINES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES MERRELL PHARMACEUTICALS INC. (US) 1996-02-29 WO disclosed