SCHEMBL7956091

SCHEMBL7956091

CCOC(=O)c1cc2c(Cl)ccc3c2n1CCCC=C3

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38
MAPK1 P28482 4/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.35
HTT P42858 2/20 0.35
ALOX15 P16050 2/20 0.35
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
TSHR P16473 2/20 0.34
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7956085 1.00 ALDH1A1 (0.39) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL7954141 0.80 MAPK1 (0.52) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL7946959 0.78 MAPK1 (0.47) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL7946984 0.77 PDE3B (0.45) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL7958065 0.76 ALDH1A1 (0.44) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL7955863 0.75 ALDH1A1 (0.41) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL7955763 0.74 ALDH1A1 (0.41) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL7954495 0.74 ALDH1A1 (0.40) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL21869100 0.71 ALDH1A1 (0.42) ALDH1A1PDE3BPDE3AMAPK1KMT2A
SCHEMBL7873755 0.70 ESR1 (0.44) ALDH1A1MAPK1GAAMAPTCYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271251-B1 CARDIOVASCULAR DISORDERS SUMITOMO PHARMACEUTICALS COMPANY LIMITED (JP) 2001-08-07 US disclosed
US-5977100-A Substituted guanidine derivatives, process for production thereof, and pharmaceutical uses thereof SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1999-11-02 US disclosed
EP-0787728-A1 Substituted guanidine derivatives, process for production thereof, and pharmaceutical uses thereof SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-08-06 EP disclosed