SCHEMBL7959142

SCHEMBL7959142

N#Cc1cccc(-c2ccc3c(c2)C(=O)CC2(CCCc4ccccc4C2)O3)c1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 9/20 0.45
PGR P06401 3/20 0.45
KDM4E B2RXH2 2/20 0.41
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.41
CHEK1 O14757 1/20 0.39
HTR2A P28223 1/20 0.39
OTUD7B Q6GQQ9 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2374444 0.95 BACE1 (0.48) BACE1PGRCHEK1HTR2AOTUD7B
SCHEMBL1821725 0.91 BACE1 (0.49) BACE1PGRKDM4EHTTATM
SCHEMBL7960189 0.91 PGR (0.51) BACE1PGRKDM4ECHEK1HTR2A
SCHEMBL7961771 0.87 PGR (0.44) BACE1PGRKDM4EHTTATM
SCHEMBL1820029 0.85 BACE1 (0.45) BACE1PGROTUD7B
SCHEMBL1820031 0.85 BACE1 (0.45) BACE1PGROTUD7B
SCHEMBL1820865 0.85 KDM4E (0.44) KDM4EHTTATM
SCHEMBL2375591 0.83 PGR (0.47) BACE1PGRCHEK1OTUD7B
SCHEMBL12246718 0.82 KDM4E (0.41) BACE1KDM4EHTTATM
SCHEMBL7949707 0.82 HDAC3 (0.52) BACE1PGRKDM4EHTTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921359-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-12-30 US disclosed
EP-2324032-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2014-10-01 EP disclosed
US-8450308-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2013-05-28 US disclosed
US-20110218192-A1 Inhibitors Of Beta-Secretase VITAE PHARMACEUTICALS, INC. (US) 2011-09-08 US disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110218192-A1 Inhibitors Of Beta-Secretase BACE1, BACE2, APP BACE1 1/4885PGR 4654/4885KDM4E 3004/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.