SCHEMBL7959792

SCHEMBL7959792

COc1cc(OC)c(NC(C)=O)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.50
CYP3A4 P08684 2/20 0.50
KDM4E B2RXH2 2/20 0.50
USP2 O75604 2/20 0.50
MAPK1 P28482 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
TP53 P04637 1/20 0.50
ALOX15 P16050 1/20 0.50
TSHR P16473 1/20 0.50
ACAT1 P24752 1/20 0.50
SOAT1 P35610 1/20 0.50
HSD17B10 Q99714 3/20 0.47
SAE1 Q9UBE0 1/20 0.47
UBA2 Q9UBT2 1/20 0.47
MEN1 O00255 1/20 0.47
PKM P14618 1/20 0.47
KMT2A Q03164 1/20 0.47
ATM Q13315 1/20 0.47
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18415560 0.86 MAPT (0.51) MAPTCYP3A4KDM4EUSP2MAPK1
SCHEMBL31465685 0.85 CYP3A4 (0.48) MAPTCYP3A4KDM4EUSP2MAPK1
SCHEMBL10683659 0.84 HSD17B10 (0.47) MAPTKDM4ESMN1; SMN2TSHRHSD17B10
SCHEMBL7959789 0.82 CYP3A4 (0.49) MAPTCYP3A4KDM4EUSP2MAPK1
SCHEMBL9641181 0.82 CYP3A4 (0.49) MAPTCYP3A4KDM4EUSP2MAPK1
SCHEMBL11271600 0.82 MAPT (0.46) MAPTKDM4EMAPK1SMN1; SMN2MEN1
SCHEMBL10676568 0.81 MAPT (0.49) MAPTCYP3A4KDM4ESMN1; SMN2HSD17B10
SCHEMBL10677501 0.81 CA12 (0.58) MAPTKDM4EMAPK1TSHRHSD17B10
SCHEMBL30977634 0.81 CYP3A4 (0.48) MAPTCYP3A4KDM4EUSP2MAPK1
SCHEMBL18415449 0.81 CYP3A4 (0.48) MAPTCYP3A4KDM4EUSP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3326715-A1 OXALIC ACID MONOAMIDE LIGAND, AND USES THEREOF IN COUPLING REACTION OF COPPER-CATALYZED ARYL HALOGEN SUBSTITUTE Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2018-05-30 EP disclosed
US-6245779-B1 ANALGESICS; ANTIINFLAMMATORY AGENTS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2001-06-12 US disclosed
EP-0997463-A1 NAPHTHYRIDINE DERIVATIVES OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2000-05-03 EP disclosed