SCHEMBL7961009

SCHEMBL7961009

Cc1ccc2c(c1)N(CC(=O)c1ccccc1C)C(=O)C(NC(=O)OC(C)(C)C)CN2C(=O)C1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 7/20 0.38
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
ACE P12821 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6176875 0.99 CCKBR (0.39) CCKBRCYP3A4MAPTTSHRACE
SCHEMBL6175171 0.93 TSHR (0.38) CCKBRMAPTTSHRACE
SCHEMBL6177673 0.92 ACE (0.38) CCKBRTSHRACE
SCHEMBL6177392 0.89 CCKBR (0.39) CCKBRCYP3A4MAPTTSHR
SCHEMBL6177871 0.89 ACE (0.39) CCKBRACE
SCHEMBL6176603 0.88 CCKBR (0.39) CCKBRCYP3A4MAPTTSHRACE
SCHEMBL7950443 0.88 CCKBR (0.39) CCKBRCYP3A4MAPTTSHRACE
SCHEMBL7959399 0.87 CCKBR (0.38) CCKBRCYP3A4MAPTTSHRACE
SCHEMBL6177504 0.87 CCKBR (0.39) CCKBRCYP3A4MAPTTSHR
SCHEMBL6178660 0.86 CCKBR (0.38) CCKBRCYP3A4MAPTTSHRACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed