SCHEMBL7962004

SCHEMBL7962004

c1ccc(-c2nccc3c2CCC3)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 4/20 0.44
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
KDM4E B2RXH2 6/20 0.43
LMNA P02545 3/20 0.43
CCR1 P32246 2/20 0.43
CCR5 P51681 2/20 0.43
CCR8 P51685 2/20 0.43
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
METAP1 P53582 1/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
DOHH Q9BU89 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
NPC1 O15118 3/20 0.42
ULK1 O75385 1/20 0.39
CDK7 P50613 1/20 0.39
CDK5 Q00535 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4052959 0.89 KDM4E (0.46) NPY5RKDM4ELMNACCR1CCR5
SCHEMBL1550749 0.79 CD44 (0.42) NPY5RKDM4ELMNACCR1CCR5
SCHEMBL18729734 0.79 NOS3 (0.47) NPY5RNOS3NOS1NOS2KDM4E
SCHEMBL5691234 0.76 NPY5R (0.51) NPY5RKDM4ELMNACCR1CCR5
SCHEMBL17702697 0.75 NOS3 (0.52) NOS3NOS1NOS2KDM4ELMNA
Ammonia Solution, Strong SCHEMBL5691104 0.75 NPY5R (0.50) NPY5RKDM4ELMNACCR1CCR5
SCHEMBL15397397 0.74 NOS3 (0.50) NOS3NOS1NOS2KDM4ELMNA
SCHEMBL15748028 0.73 KDM4E (0.48) KDM4ELMNACCR1CCR5CCR8
SCHEMBL3367025 0.72 NPY5R (0.48) NPY5RNOS3NOS1NOS2KDM4E
SCHEMBL19373744 0.71 NOS3 (0.47) NOS3NOS1NOS2KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313305-B1 ANTIBIOTICS, BACTERICIDES HOECHST MARION ROUSSEL (FR) 2001-11-06 US disclosed
US-5883248-A QUATERNARY AMMONIUM INTERMEDIATES ROUSSEL UCLAF (FR) 1999-03-16 US disclosed
US-5763617-A Cephalosporins ROUSSEL UCLAF (FR) 1998-06-09 US disclosed
US-5728828-A A 3-(3-CHLORO- OR IODOPROP-1-EN-1-YL),7-(2-AMINOTHIAZOL-4-YL) ((CARBOXY)(PHENYL)METHOXYIMINO)ACETAMIDO-3-CEPHEM; GRAMNEGATIVE AND -POSITIVE BACTERIA, ESP. ANTIBIOTIC-RESISTANCE STAPHYLOCOCCUS ROUSSEL UCLAF (FR) 1998-03-17 US disclosed
US-5712266-A Cephalosporins ROUSSEL UCLAF (FR) 1998-01-27 US disclosed
US-5587372-A BACERICIDES ROUSSEL UCLAF (FR) 1996-12-24 US disclosed