SCHEMBL7962148

SCHEMBL7962148

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCC(C=O)N2CCN(C)CC2)ccc1NC(=O)c1cccc2ncn(C)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.34
MAP3K7 O43318 4/20 0.33
EGFR P00533 1/20 0.33
KDR P35968 1/20 0.33
FLT3 P36888 1/20 0.33
CYP3A4 P08684 1/20 0.33
LPAR1 Q92633 1/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
HCN1 O60741 1/20 0.32
HCN4 Q9Y3Q4 1/20 0.32
AVPR2 P30518 1/20 0.32
AVPR1A P37288 1/20 0.32
AVPR1B P47901 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPK14 Q16539 1/20 0.31
CCNK O75909 1/20 0.31
CCNA2 P20248 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7424661 0.99 IRAK4 (0.33) IRAK4MAP3K7EGFRKDRFLT3
SCHEMBL7420333 0.88 CYP3A4 (0.34) IRAK4MAP3K7EGFRCYP3A4LPAR1
SCHEMBL7964976 0.86 AVPR2 (0.39) IRAK4MAP3K7FLT3LPAR1AVPR2
SCHEMBL7594829 0.86 MAP3K7 (0.34) IRAK4MAP3K7CYP3A4LPAR1ADRA1D
Hydrochloric Acid SCHEMBL7965268 0.86 AVPR2 (0.39) IRAK4MAP3K7FLT3LPAR1AVPR2
Hydrochloric Acid SCHEMBL7971987 0.86 MAP3K7 (0.39) MAP3K7
SCHEMBL7975460 0.86 MAP3K7 (0.34) IRAK4MAP3K7ADRA1DADRA1AADRA1B
SCHEMBL7476561 0.85 PTK2 (0.36) IRAK4MAP3K7ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7335533 0.85 ABCB1 (0.34) IRAK4MAP3K7CYP3A4LPAR1ADRA1D
SCHEMBL7964805 0.85 MAP3K7 (0.33) IRAK4MAP3K7CYP3A4LPAR1ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed