SCHEMBL7420333

SCHEMBL7420333

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCC(C=O)N2CCN(C)CC2)ccc1NC(=O)c1cccc(N)c1N

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.34
LPAR1 Q92633 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
ADRA1B P35368 2/20 0.34
MAP3K7 O43318 4/20 0.33
HCN1 O60741 1/20 0.33
HCN4 Q9Y3Q4 1/20 0.33
AVPR2 P30518 2/20 0.33
AVPR1A P37288 2/20 0.33
AVPR1B P47901 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ABCB1 P08183 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
EGFR P00533 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7966897 0.92 ALDH1A1 (0.34) CYP3A4KMT2AABCB1ABCG2EGFR
SCHEMBL7594829 0.88 MAP3K7 (0.34) CYP3A4LPAR1IRAK4ADRA1DADRA1A
SCHEMBL7476561 0.88 PTK2 (0.36) IRAK4ADRA1DADRA1AADRA1BMAP3K7
SCHEMBL7962148 0.88 IRAK4 (0.34) CYP3A4LPAR1IRAK4ADRA1DADRA1A
Hydrochloric Acid SCHEMBL7469087 0.88 MAP3K7 (0.34) IRAK4ADRA1DADRA1AADRA1BMAP3K7
SCHEMBL7346091 0.87 HCN1 (0.35) CYP3A4LPAR1ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7424661 0.87 IRAK4 (0.33) CYP3A4LPAR1IRAK4ADRA1DADRA1A
Hydrochloric Acid SCHEMBL7335533 0.87 ABCB1 (0.34) CYP3A4LPAR1IRAK4ADRA1DADRA1A
SCHEMBL7978086 0.87 MAP3K7 (0.32) CYP3A4LPAR1IRAK4ADRA1DADRA1A
SCHEMBL7429725 0.87 MAP3K7 (0.33) IRAK4ADRA1DADRA1AADRA1BMAP3K7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed
EP-0946519-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-06 EP disclosed
WO-1998024771-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-06-11 WO disclosed