SCHEMBL7963215

SCHEMBL7963215

CCCCC(C)(CC(=O)OC)c1nc(C)nc2c1c(SC)nn2-c1c(Cl)cc(Cl)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 18/20 0.46
CCND1 P24385 18/20 0.46
CCNE2 O96020 11/20 0.45
CCNE1 P24864 11/20 0.45
CDK2 P24941 11/20 0.45
CCNB2 O95067 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
CRHR1 P34998 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8112963 0.89 CDK4 (0.45) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7962973 0.85 CDK4 (0.49) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7964093 0.83 CDK4 (0.51) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7965540 0.81 CRHR1 (0.49) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7962975 0.80 CDK4 (0.47) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7952791 0.77 CDK4 (0.47) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7953100 0.72 CDK4 (0.63) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL5600331 0.71 CDK4 (0.53) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7965911 0.70 CRHR1 (0.63) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7953286 0.70 CDK4 (0.46) CDK4CCND1CCNE2CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6218397-B1 FOR THERAPY OF STRESS-RELATED ILLNESSES, SUCH AS STRESS-INDUCED DEPRESSION, ANXIETY, AND HEADACHE; ABDOMINAL BOWEL SYNDROME; INFLAMMATORY DISEASES; IMMUNE SUPPRESSION; ALZHEIMER'S DISEASE; GASTRONINTESTINAL DISEASES PFIZER INC 2001-04-17 US disclosed