SCHEMBL7964324

SCHEMBL7964324

CCN(CC)C(=O)c1ccc(Cl)nc1-c1ccccc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
HPGD P15428 3/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HCRTR1 O43613 4/20 0.40
HCRTR2 O43614 4/20 0.40
GHSR Q92847 1/20 0.38
ALDH1A1 P00352 3/20 0.38
LMNA P02545 1/20 0.38
GPBAR1 Q8TDU6 2/20 0.38
PDE5A O76074 1/20 0.37
CYP3A4 P08684 1/20 0.37
PDE4A P27815 1/20 0.37
PDE6C P51160 1/20 0.37
PDE7A Q13946 1/20 0.37
PDE11A Q9HCR9 1/20 0.37
PDE10A Q9Y233 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12329757 0.76 MEN1 (0.48) KEAP1TSHRMAPK1HPGDNPC1
SCHEMBL7110905 0.75 GPBAR1 (0.53) KEAP1TSHRMAPK1HPGDNPC1
SCHEMBL14134227 0.75 TSHR (0.58) KEAP1TSHRMAPK1HPGDNPC1
SCHEMBL14052388 0.73 KEAP1 (0.51) KEAP1TSHRMAPK1HPGDNPC1
SCHEMBL150008 0.71 TSHR (0.75) KEAP1TSHRMAPK1HPGDSMN1; SMN2
SCHEMBL18564898 0.71 ADORA2A (0.42) TSHRMAPK1HPGDNPC1RAB9A
SCHEMBL29381824 0.71 TSHR (0.75) KEAP1TSHRMAPK1HPGDSMN1; SMN2
SCHEMBL4467948 0.69 TSHR (0.54) KEAP1TSHRMAPK1HPGDSMN1; SMN2
SCHEMBL14529999 0.68 TSHR (0.47) KEAP1TSHRMAPK1HPGDNPC1
Hydrochloric Acid SCHEMBL813914 0.68 TSHR (0.53) KEAP1TSHRMAPK1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303790-B1 REACTING SUBSTITUTED NICOTINAMIDE WITH GRIGNARD REAGENT, OXIDIZING PRODUCT, REACTING WITH HALO-SUBSTITUTED AROMATIC COMPOUND HOFFMAN-LA ROCHE INC. 2001-10-16 US disclosed