SCHEMBL7964584

SCHEMBL7964584

Bc1ccc2c(c1)C1(CC(c3ccccc3F)O2)N=C(SC)N(C)C1=O

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
BACE1 P56817 10/20 0.33
CTSD P07339 8/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7961006 0.93 BACE1 (0.33) BACE1CTSD
SCHEMBL2376169 0.89 BACE1 (0.40) KDM4EALDH1A1GAAMAPTALOX15
SCHEMBL7958172 0.87 BACE1 (0.43) BACE1CTSD
SCHEMBL7960450 0.85 BACE1 (0.37) BACE1CTSD
SCHEMBL2375720 0.82 BACE1 (0.39) BACE1CTSD
SCHEMBL7950191 0.81 BACE1 (0.38) BACE1CTSD
SCHEMBL16136547 0.79 BACE1 (0.41) BACE1CTSD
SCHEMBL7961021 0.78 BACE1 (0.32) BACE1
SCHEMBL2377481 0.76 MAOB (0.43) BACE1CTSD
SCHEMBL2375751 0.76 BACE1 (0.55) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed