SCHEMBL7964773

SCHEMBL7964773

O=C(O)c1ccc(C(=O)N2CCN(C(=O)N3CCOCC3)CC2)cc1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.79
AKR1C3 P42330 2/20 0.74
HPGD P15428 4/20 0.64
PHGDH O43175 1/20 0.63
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
ALDH1A1 P00352 4/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
MAPK1 P28482 1/20 0.55
KDM4E B2RXH2 1/20 0.55
MAPT P10636 1/20 0.55
HTT P42858 1/20 0.55
USP2 O75604 1/20 0.54
POLB P06746 1/20 0.54
DNMT1 P26358 1/20 0.54
PTPN7 P35236 1/20 0.54
KMT2A Q03164 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
PKM P14618 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696938 0.93 HPGD (0.72) TSHRAKR1C3HPGDPHGDHALDH1A1
SCHEMBL10720943 0.86 PHGDH (0.81) TSHRAKR1C3HPGDPHGDHALDH1A1
SCHEMBL9133746 0.84 ALDH1A1 (0.64) TSHRHPGDALDH1A1SMN1; SMN2MAPK1
SCHEMBL946143 0.80 HPGD (0.86) TSHRAKR1C3HPGDPHGDHALDH1A1
SCHEMBL28296651 0.80 HPGD (0.86) TSHRAKR1C3HPGDPHGDHALDH1A1
Ammonia Solution, Strong SCHEMBL6028542 0.79 HPGD (0.83) TSHRAKR1C3HPGDPHGDHALDH1A1
SCHEMBL2199279 0.79 PHGDH (0.71) TSHRAKR1C3HPGDPHGDHALDH1A1
SCHEMBL30449295 0.79 HPGD (0.83) TSHRAKR1C3HPGDPHGDHALDH1A1
SCHEMBL8150805 0.78 HPGD (0.76) TSHRHPGDPHGDHALDH1A1SMN1; SMN2
SCHEMBL27045664 0.78 HPGD (1.00) TSHRAKR1C3HPGDPHGDHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265381-B1 MORPHOLINOUREA AND RELATED DERIVATIVES OF PENTAFLUOROETHYL PEPTIDES MERRELL PHARMACEUTICALS, INC. 2001-07-24 US disclosed