SCHEMBL7965589

SCHEMBL7965589

CC(C)(C)OC(=O)Nc1nnc(-c2ccccc2)n(CC(=O)O)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD9 Q9H8M2 1/20 0.43
CNR2 P34972 1/20 0.41
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
BRD4 O60885 2/20 0.40
HSD17B10 Q99714 1/20 0.39
GAA P10253 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ELANE P08246 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA7 P43166 1/20 0.37
CA14 Q9ULX7 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7960757 0.83 CNR2 (0.43) BRD9CNR2KDM4EHPGDHSD17B10
SCHEMBL7953847 0.81 ELANE (0.53) BRD9CNR2ELANE
SCHEMBL8325921 0.72 HDAC6 (0.39) BRD9CNR2BRD4CA12CA1
SCHEMBL7964912 0.72 CNR2 (0.41) BRD9CNR2KDM4EHPGDHSD17B10
SCHEMBL14548656 0.71 ELANE (0.47) BRD9CNR2ELANE
SCHEMBL7959556 0.70 CNR2 (0.40) BRD9CNR2KDM4EALDH1A1AKT1
SCHEMBL3495412 0.70 BRD4 (0.48) BRD9BRD4CYP1A2CYP2C9CYP2C19
SCHEMBL3816887 0.69 DRD2 (0.46) BRD4AKT1
SCHEMBL5848201 0.68 F7 (0.52) BRD4
SCHEMBL6163930 0.68 F7 (0.52) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271238-B1 USEFUL IN TREATING AND PREVENTING DISEASES INVOLVING CHYMOTRYPSIN TYPE PROTEASES WHICH ARE RELATED TO ASTHMA, ALLERGY, INFLAMMATIONS, RHEUMATISM, HYPERTENSION, HEART FAILURE, MYOCARDIAL INFARCTION, AND CARDIAC HYPERTROPHY NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-08-07 US disclosed