SCHEMBL7965941

SCHEMBL7965941

CC(C)(C)Oc1cccc2[nH]c(C3CCNCC3)nc12

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.54
PARP2 Q9UGN5 3/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
CDK1 P06493 1/20 0.38
CDK9 P50750 1/20 0.38
HTR2C P28335 2/20 0.38
JUND P17535 1/20 0.37
FOSB P53539 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7966174 0.82 PARP1 (0.54) PARP1PARP2CDK1CDK9
SCHEMBL7965946 0.80 CDK1 (0.40) PARP1CDK1CDK9HTR2CJUND
SCHEMBL7215446 0.78 PARP1 (0.61) PARP1PARP2ALDH1A1POLBMAPT
SCHEMBL6872238 0.78 PARP1 (0.68) PARP1PARP2
SCHEMBL7956612 0.77 PARP1 (0.57) PARP1PARP2ALDH1A1POLBMAPT
SCHEMBL5201219 0.76 PARP1 (0.55) PARP1PARP2ALDH1A1POLBMAPT
SCHEMBL6871409 0.76 PARP1 (0.56) PARP1PARP2
SCHEMBL6129581 0.75 PARP1 (0.65) PARP1PARP2ALDH1A1POLBMAPT
SCHEMBL6872911 0.75 PARP1 (0.61) PARP1PARP2
SCHEMBL3972140 0.74 PARP1 (0.49) PARP1PARP2ALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303627-B1 FOR THERAPY OF PHYSIOLOGICAL AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY 2001-10-16 US disclosed
EP-0965587-A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1999-12-22 EP disclosed