SCHEMBL7966971

SCHEMBL7966971

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCC(=C=O)N2CCN(C)CC2)ccc1C(=O)Nc1cccc2[nH]c(CN3CCOCC3)nc12

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 2/20 0.34
PDCD1 Q15116 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
MAPK14 Q16539 1/20 0.33
KDR P35968 2/20 0.33
EGFR P00533 1/20 0.33
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HDAC1 Q13547 1/20 0.32
FGFR3 P22607 1/20 0.32
DYRK1A Q13627 1/20 0.32
ALK Q9UM73 1/20 0.32
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7964608 0.96 ALK (0.34) KDREGFRHDAC1FGFR3ALK
Hydrochloric Acid SCHEMBL7472559 0.96 ALK (0.34) KDREGFRHDAC1FGFR3ALK
SCHEMBL7967130 0.95 CACNA1G (0.33) HDAC1ALK
SCHEMBL7954417 0.95 MLLT1 (0.34) ALDH1A1LMNAHDAC1ALK
SCHEMBL7485529 0.94 IRAK4 (0.36) CD274PDCD1IRAK4MAPK14KDR
SCHEMBL7966975 0.93 KDM4E (0.35) CD274PDCD1IRAK4MAPK14KDR
Hydrochloric Acid SCHEMBL7978179 0.93 KDM4E (0.35) CD274PDCD1IRAK4MAPK14KDR
SCHEMBL7964677 0.92 HDAC3 (0.34) KDREGFRHDAC1
SCHEMBL7480416 0.91 ABCB1 (0.34) KDREGFRHDAC1
Hydrochloric Acid SCHEMBL7963051 0.91 HDAC3 (0.34) KDREGFRHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316482-B1 FOR THERAPY AND PROPHYLAXIS OF HYPERTENSION, HEART FAILURE, RENAL INSUFFICIENCY, EDEMA, ASCITES, VASOPRESSIN PARASECRETION SYNDROME, HEPATOCIRRHOSIS, HYPONATREMIA, HYPOKALEMIA, DIABETIC, CIRCULATION DISORDER, CEREBROVASCULAR DISEASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed