SCHEMBL7971348

SCHEMBL7971348

COc1ccc(CC(NC(=O)OCc2ccccc2)C(=O)NNC(=O)c2ccccc2)cc1

nearest known ligand 0.83

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.83
CTSK P43235 7/20 0.64
HDAC8 Q9BY41 2/20 0.61
F2 P00734 1/20 0.61
ALDH1A1 P00352 2/20 0.59
CTSL P07711 2/20 0.58
CTSS P25774 2/20 0.58
CTSB P07858 1/20 0.57
ATM Q13315 1/20 0.56
ALOX15 P16050 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971421 0.91 TACR1 (1.00) TACR1CTSKALDH1A1CTSLCTSS
SCHEMBL7970040 0.90 TACR1 (0.67) TACR1CTSKHDAC8F2CTSL
SCHEMBL8118400 0.88 TACR1 (0.61) TACR1CTSKHDAC8ALDH1A1CTSL
SCHEMBL10706786 0.86 HDAC8 (0.68) TACR1CTSKHDAC8F2CTSL
SCHEMBL7970037 0.86 HDAC8 (0.65) TACR1CTSKHDAC8F2ALDH1A1
SCHEMBL14684392 0.85 HDAC8 (0.64) TACR1CTSKHDAC8F2CTSL
SCHEMBL7317573 0.85 HDAC8 (0.64) TACR1CTSKHDAC8F2CTSL
SCHEMBL8569421 0.85 ALDH1A1 (0.65) TACR1CTSKHDAC8F2ALDH1A1
SCHEMBL7044299 0.85 ATM (0.67) CTSKHDAC8F2ALDH1A1CTSL
SCHEMBL9716778 0.85 ATM (0.67) CTSKHDAC8F2ALDH1A1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6172108-B1 NEUROPEPTIDE Y RECEPTOR LIGANDS; TREATING PSYCHOLOGICAL, EATING, SLEEP, AND SEXUAL DISORDERS; HYPOTENSIVE, ANXIOLYTIC, ANTIDEPRESSANT, AND ANTIDIABETIC AGENTS ADIR ET COMPAGNIE (FR) 2001-01-09 US disclosed