SCHEMBL7972075

SCHEMBL7972075

CCOC(=O)CCc1ccc(NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.56
CYP4A11 Q02928 1/20 0.56
CYP17A1 P05093 1/20 0.51
CYP4Z1 Q86W10 1/20 0.49
PPARG P37231 2/20 0.48
PPARA Q07869 1/20 0.48
DRD2 P14416 1/20 0.48
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MITF O75030 1/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.46
PPID Q08752 1/20 0.45
NAMPT P43490 2/20 0.44
EPHX2 P34913 1/20 0.43
MAPK14 Q16539 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
NCOR2 Q9Y618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6755422 0.87 CYP17A1 (0.54) CYP17A1PPARGPPARADRD2LMNA
SCHEMBL15709727 0.86 LMNA (0.62) CYP17A1CYP4Z1PPARGPPARALMNA
SCHEMBL7421780 0.85 MAPT (0.47) CYP4F2CYP4A11LMNAMAPTSMN1; SMN2
SCHEMBL4495406 0.84 CYP4F2 (0.56) CYP4F2CYP4A11CYP4Z1MAPTSMN1; SMN2
SCHEMBL6376720 0.84 CYP4F2 (0.56) CYP4F2CYP4A11CYP4Z1MAPTSMN1; SMN2
SCHEMBL1000732 0.83 NR1H4 (0.58) CYP17A1PPARGPPARADRD2PTGDR2
SCHEMBL12677009 0.83 CYP17A1 (0.58) CYP17A1PPARGPPARADRD2PTGDR2
SCHEMBL3173008 0.83 PPARG (0.53) CYP17A1PPARGPPARADRD2LMNA
SCHEMBL23513700 0.82 CA12 (0.46) CYP4F2CYP4A11CYP17A1PPARGLMNA
SCHEMBL6984766 0.81 CYP4F2 (0.64) CYP4F2CYP4A11CYP4Z1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235731-B1 REDUCING BLOOD LIPIDS, SUGARS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
CN-1223659-A Fused imidazopyridine derivatives as antihyperlipidemic agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-07-21 CN disclosed
EP-0915888-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS Takeda Chemical Industries, Ltd. (JP) 1999-05-19 EP disclosed
WO-1997040051-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-30 WO disclosed