SCHEMBL797279

SCHEMBL797279

CCCC(C(=O)O)=C(CC)CCN

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.41
GRIA4 P48058 1/20 0.41
GRIK3 Q13003 1/20 0.41
GRIK5 Q16478 1/20 0.41
FFAR3 O14843 4/20 0.37
HDAC3 O15379 4/20 0.37
HDAC1 Q13547 4/20 0.37
HDAC2 Q92769 4/20 0.37
HDAC8 Q9BY41 4/20 0.37
ALDH1A1 P00352 1/20 0.34
FNTA P49354 2/20 0.34
FNTB P49356 2/20 0.34
THRB P10828 2/20 0.34
PGGT1B P53609 1/20 0.34
CES2 O00748 2/20 0.33
CES1 P23141 2/20 0.33
CTSD P07339 1/20 0.32
TSHR P16473 2/20 0.31
GABRR3 A8MPY1 1/20 0.30
GABRP O00591 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methacrylic Acid SCHEMBL29514865 0.91 GRIK1 (0.36) GRIK1GRIA4GRIK3GRIK5FFAR3
SCHEMBL4592350 0.85 GRIK1 (0.50) GRIK1GRIA4GRIK3GRIK5FFAR3
SCHEMBL9747819 0.84 GRIK1 (0.48) GRIK1GRIA4GRIK3GRIK5FFAR3
SCHEMBL8599484 0.79 FNTA (0.52) ALDH1A1FNTAFNTBTHRBPGGT1B
SCHEMBL8599489 0.79 FNTA (0.52) ALDH1A1FNTAFNTBTHRBPGGT1B
SCHEMBL28065698 0.78 FFAR3 (0.43) GRIK1GRIA4GRIK3GRIK5FFAR3
SCHEMBL31195898 0.77 HDAC3 (0.48) GRIK1GRIA4GRIK3GRIK5FFAR3
SCHEMBL9158350 0.77 GRIK1 (0.47) GRIK1GRIA4GRIK3GRIK5FFAR3
SCHEMBL3917513 0.75 CYP2D6 (0.48) GRIK1GRIA4GRIK3GRIK5HDAC3
SCHEMBL554602 0.74 HDAC3 (0.56) FFAR3HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0952195-B1 Ink set for improved print quality HEWLETT PACKARD CO (US) 2003-06-25 EP claimed
EP-0952196-B1 Ink-jet printing system for improved print quality HEWLETT PACKARD CO (US) 2003-06-25 EP claimed
EP-1299458-B1 AQUEOUS DISPERSION COMPRISING VISCOUS SILICONE OILS CROSSLINKABLE BY CONDENSATION INTO AN ADHERING ELASTOMER FOR USE AS SEALANTS OR PAINTS AND PREPARATION METHOD HENKEL AG & CO KGAA (DE) 2011-11-30 EP disclosed
EP-1406979-B1 METHOD FOR PRODUCTION OF A SEALED COATING FOR SURFACES OF BUILDINGS COMPRISING A CROSS-LINKED SEALED SILICONE MEMBRANE, ADHESIVE AND READY-TO-USE KIT FOR APPLICATION OF SAID METHOD HENKEL AG & CO KGAA (DE) 2011-05-25 EP disclosed
US-7001616-B2 Microspheres for use in the treatment of cancer UNIVERSITY OF FLORIDA (US) 2006-02-21 US disclosed
EP-1406979-A1 METHOD FOR PRODUCTION OF A SEALED COATING FOR SURFACES OF BUILDINGS COMPRISING A CROSS-LINKED SEALED SILICONE MEMBRANE, ADHESIVE AND READY-TO-USE KIT FOR APPLICATION OF SAID METHOD Rhodia Chimie (FR) 2004-04-14 EP disclosed
US-20030202936-A1 Microspheres for use in the treatment of cancer FLORIDA, UNIVERSITY OF 2003-10-30 US disclosed
EP-0885254-B1 COMPOSITE PARTICLES INCLUDING AN ORGANIC POLYMER AND AN OXIDE AND/OR HYDROXIDE RHODIA CHIMIE SA (FR) 2003-08-13 EP disclosed
US-6602524-B2 Ph sensitivie spheres; crosslinked polymer; drug delivery UNIVERSITY OF FLORIDA 2003-08-05 US disclosed
EP-1299458-A1 AQUEOUS DISPERSION BASED OF VISCOUS SILICONE OILS CROSSLINKABLE BY CONDENSATION INTO AN ADHERING ELASTOMER FOR USE IN PARTICULAR AS SEALANTS OR PAINTS, PREPARATION METHOD Rhodia Chimie (FR) 2003-04-09 EP disclosed
WO-2003002677-A1 METHOD FOR PRODUCTION OF A SEALED COATING FOR SURFACES OF BUILDINGS COMPRISING A CROSS-LINKED SEALED SILICONE MEMBRANE, ADHESIVE AND READY-TO-USE KIT FOR APPLICATION OF SAID METHOD RHODIA CHIMIE (FR) 2003-01-09 WO disclosed
US-20020009415-A1 Microspheres for use in the treatment of cancer FLORIDA, UNIVERSITY OF 2002-01-24 US disclosed
WO-2002000770-A1 AQUEOUS DISPERSION BASED OF VISCOUS SILICONE OILS CROSSLINKABLE BY CONDENSATION INTO AN ADHERING ELASTOMER FOR USE IN PARTICULAR AS SEALANTS OR PAINTS, PREPARATION METHOD RHODIA CHIME (FR) 2002-01-03 WO disclosed
US-6136891-A ORGANIC POLYMER CORE AND METAL OXIDE COATING, FILLERS OR ADDITIVES FOR PLASTICS OR ELASTOMERS. RHODIA CHIMIE (FR) 2000-10-24 US disclosed
CN-1236793-A Ink set for improved print quality HEWLETT PACKARD CO (US) 1999-12-01 CN disclosed
CN-1236794-A Ink-jet printing system for improved print quality HEWLETT PACKARD CO (US) 1999-12-01 CN disclosed
EP-0885254-A1 COMPOSITE PARTICLES INCLUDING AN ORGANIC POLYMER AND AN OXIDE AND/OR HYDROXIDE RHODIA CHIMIE (FR) 1998-12-23 EP disclosed
WO-1997032920-A1 COMPOSITE PARTICLES INCLUDING AN ORGANIC POLYMER AND AN OXIDE AND/OR HYDROXIDE RHODIA CHIMIE (FR) 1997-09-12 WO disclosed
EP-0699703-A1 Composite and hollow particles of calcium carbonate RHONE-POULENC CHIMIE (FR) 1996-03-06 EP disclosed