SCHEMBL7973580

SCHEMBL7973580

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCN(C)CC2)ccc1C(=O)Nc1cccc2[nH]c(C(=O)N(C)C)nc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 3/20 0.34
AVPR1A P37288 3/20 0.34
AVPR1B P47901 2/20 0.34
IRAK4 Q9NWZ3 2/20 0.34
MAP3K7 O43318 4/20 0.34
AURKA O14965 1/20 0.33
JAK2 O60674 1/20 0.33
LCK P06239 1/20 0.33
LYN P07948 1/20 0.33
KIT P10721 1/20 0.33
TYK2 P29597 1/20 0.33
TEC P42680 1/20 0.33
TXK P42681 1/20 0.33
BMX P51813 1/20 0.33
BTK Q06187 1/20 0.33
ITK Q08881 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7962022 0.99 AVPR2 (0.34) AVPR2AVPR1AAVPR1BIRAK4MAP3K7
SCHEMBL7480849 0.94 AVPR2 (0.35) AVPR2AVPR1AAVPR1BIRAK4MAP3K7
Hydrochloric Acid SCHEMBL7481449 0.93 AVPR2 (0.35) AVPR2AVPR1AAVPR1BIRAK4MAP3K7
SCHEMBL7480376 0.93 AVPR2 (0.38) AVPR2AVPR1AAVPR1BIRAK4MAP3K7
Dimethylamine SCHEMBL7972125 0.93 AVPR2 (0.35) AVPR2AVPR1AAVPR1BIRAK4MAP3K7
SCHEMBL7964762 0.93 AVPR2 (0.37) AVPR2AVPR1AAVPR1BIRAK4MAP3K7
SCHEMBL7480014 0.92 MAP3K7 (0.32) IRAK4MAP3K7AURKAJAK2LCK
Hydrochloric Acid SCHEMBL7597564 0.92 AVPR2 (0.37) AVPR2AVPR1AAVPR1BIRAK4MAP3K7
SCHEMBL7481684 0.92 AVPR2 (0.34) AVPR2AVPR1AAVPR1BIRAK4MAP3K7
SCHEMBL7962954 0.92 AVPR2 (0.34) AVPR2AVPR1AAVPR1BIRAK4MAP3K7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed