SCHEMBL7973583

SCHEMBL7973583

CCCN(Cc1ccccc1)C(C)CCC(C#N)(c1ccc(Br)cc1)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.46
EBP Q15125 2/20 0.46
BCHE P06276 2/20 0.43
OPRM1 P35372 3/20 0.34
OPRK1 P41145 2/20 0.34
TSHR P16473 5/20 0.33
CYP2C19 P33261 3/20 0.33
KCNH2 Q12809 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
SLC22A1 O15245 2/20 0.33
CHRM2 P08172 2/20 0.33
HTR1A P08908 2/20 0.33
ADRA2A P08913 2/20 0.33
DRD2 P14416 2/20 0.33
ADRA2B P18089 2/20 0.33
ADRA2C P18825 2/20 0.33
DRD1 P21728 2/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
ADRA1A P35348 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968805 0.92 SIGMAR1 (0.47) SIGMAR1EBPBCHEOPRM1OPRK1
SCHEMBL7965942 0.91 SIGMAR1 (0.45) SIGMAR1EBPBCHEOPRM1OPRK1
SCHEMBL7973937 0.90 SIGMAR1 (0.44) SIGMAR1EBPBCHEOPRM1OPRK1
SCHEMBL7968643 0.89 SIGMAR1 (0.46) SIGMAR1EBPBCHEOPRM1OPRK1
SCHEMBL7971672 0.89 SIGMAR1 (0.46) SIGMAR1EBPBCHEOPRM1OPRK1
SCHEMBL7974380 0.89 SIGMAR1 (0.46) SIGMAR1EBPBCHEOPRM1OPRK1
SCHEMBL7970398 0.89 SIGMAR1 (0.41) SIGMAR1EBPBCHEOPRM1OPRK1
SCHEMBL7969033 0.86 SIGMAR1 (0.57) SIGMAR1EBPOPRM1OPRK1TSHR
SCHEMBL7970967 0.85 BCHE (0.43) SIGMAR1EBPBCHEOPRM1OPRK1
SCHEMBL7973615 0.85 BCHE (0.43) SIGMAR1EBPBCHEOPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed