SCHEMBL7974939

SCHEMBL7974939

NC(=O)c1ccc2nc(-c3[nH]nc(-c4ccc(CN5CCOCC5)cc4)c3O)[nH]c2c1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.59
HDAC3 O15379 2/20 0.59
HDAC1 Q13547 2/20 0.59
HDAC2 Q92769 2/20 0.59
HDAC8 Q9BY41 2/20 0.59
CHEK1 O14757 2/20 0.55
CDK7 P50613 1/20 0.54
F9 P00740 1/20 0.53
F10 P00742 1/20 0.53
F11 P03951 1/20 0.53
F7 P08709 1/20 0.53
CHEK2 O96017 11/20 0.51
AURKA O14965 2/20 0.50
CDK1 P06493 2/20 0.50
CCNB1 P14635 2/20 0.50
CDK2 P24941 2/20 0.50
AURKB Q96GD4 2/20 0.50
PARP1 P09874 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20307778 0.91 HDAC6 (0.57) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL7970994 0.84 HDAC6 (0.59) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL10139860 0.83 F9 (0.69) CHEK1F9F10F11F7
SCHEMBL7959397 0.82 CHEK2 (0.68) F9F10F11F7CHEK2
SCHEMBL7972717 0.80 F9 (0.77) CHEK1F9F10F11F7
SCHEMBL10172686 0.80 CHEK2 (0.69) F9F10F11F7CHEK2
SCHEMBL10139859 0.77 CHEK2 (0.64) F9F10F11F7CHEK2
SCHEMBL10139999 0.76 HDAC6 (0.54) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL18229535 0.76 HDAC6 (0.98) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL20307772 0.76 F9 (0.64) F9F10F11F7CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed