SCHEMBL7959397

SCHEMBL7959397

NC(=O)c1ccc2nc(-c3[nH]nc(-c4ccc(Cl)cc4)c3O)[nH]c2c1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 19/20 0.68
F9 P00740 1/20 0.64
F10 P00742 1/20 0.64
F11 P03951 1/20 0.64
F7 P08709 1/20 0.64
MEN1 O00255 1/20 0.62
THRB P10828 1/20 0.62
KMT2A Q03164 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10139860 0.93 F9 (0.69) CHEK2F9F10F11F7
SCHEMBL7972721 0.90 CHEK2 (0.67) CHEK2F9F10F11F7
SCHEMBL10172686 0.89 CHEK2 (0.69) CHEK2F9F10F11F7
SCHEMBL7972717 0.89 F9 (0.77) CHEK2F9F10F11F7
SCHEMBL20307772 0.89 F9 (0.64) CHEK2F9F10F11F7
SCHEMBL10139859 0.87 CHEK2 (0.64) CHEK2F9F10F11F7
SCHEMBL20307778 0.83 HDAC6 (0.57) CHEK2F9F10F11F7
SCHEMBL7978282 0.83 CHEK2 (0.56) CHEK2F9F10F11F7
SCHEMBL7974939 0.82 HDAC6 (0.59) CHEK2F9F10F11F7
SCHEMBL7972817 0.81 F9 (0.54) CHEK2F9F10F11F7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2805939-B1 Heterocyclic compounds as factor IXA inhibitors. MERCK SHARP & DOHME (US) 2018-06-27 EP disclosed
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed