SCHEMBL7974979

SCHEMBL7974979

CN(Cc1ccc(NC(=O)C2=Cc3cc(-c4ccc(OC(F)(F)F)cc4)ccc3S(=O)(=O)CC2)cc1)C1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.58
CCR5 P51681 15/20 0.46
CXCR3 P49682 3/20 0.41
CCR7 P32248 2/20 0.41
CXCR5 P32302 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7972718 0.91 CCR2 (0.61) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7958720 0.91 CCR2 (0.61) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7958790 0.90 CCR2 (0.64) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7975101 0.90 CCR2 (0.64) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7928215 0.90 CCR2 (0.60) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7969655 0.90 CCR2 (0.60) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7968984 0.90 CCR2 (0.60) CCR2CCR5CXCR3CCR7CXCR5
Hydrochloric Acid SCHEMBL7975094 0.89 CCR2 (0.59) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7968833 0.89 CCR2 (0.61) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7958933 0.89 CCR2 (0.61) CCR2CCR5CXCR3CCR7CXCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed