SCHEMBL7975987

SCHEMBL7975987

COc1cc(Cc2csc3cc(OCc4ccccc4-c4ccc(N)cc4)ccc23)ccc1CN1CCCC1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 8/20 0.51
F2 P00734 10/20 0.48
HTR7 P34969 1/20 0.40
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7355874 0.81 CD274 (0.54) CD274F2HRH3
SCHEMBL6173777 0.79 F2 (0.67) CD274F2
SCHEMBL7446083 0.75 F2 (0.60) CD274F2HRH3
SCHEMBL7348647 0.74 F2 (0.53) CD274F2HRH3
SCHEMBL7447052 0.73 CD274 (0.55) CD274F2HRH3
SCHEMBL6172550 0.73 F2 (0.76) CD274F2
SCHEMBL6173290 0.73 ESR1 (0.52) F2
SCHEMBL7353107 0.73 HRH3 (0.48) CD274F2HRH3
SCHEMBL7452057 0.72 HRH3 (0.54) CD274F2HRH3
SCHEMBL6172092 0.71 F2 (0.73) CD274F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288105-B1 COMPOUNDS SUCH AS (S)-2-(4-((2-AMINO-3-HYDROXY-1-OXOPROPYL)AMINO)PHENYL)-6-HYDRO XY-3-(3-METHOXY-4-(1-PYRROLIDINYLMETHYL)BENZYL)BENZO(B)THIOPHE NE ELI LILLY AND COMPANY 2001-09-11 US disclosed