SCHEMBL7977375

SCHEMBL7977375

CN1CCCc2cnccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.49
CHRM3 P20309 2/20 0.49
CHRM1 P11229 1/20 0.49
SIGMAR1 Q99720 1/20 0.48
CHRM4 P08173 1/20 0.48
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP3A4 P08684 2/20 0.39
NPSR1 Q6W5P4 1/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31555114 1.00 CHRM2 (0.49) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL22674240 0.95 SIGMAR1 (0.52) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL256358 0.89 CYP3A4 (0.46) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL31518333 0.89 CYP3A4 (0.46) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL16998410 0.85 SIGMAR1 (0.48) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL22674242 0.80 SIGMAR1 (0.52) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL22313609 0.78 CHRM2 (0.49) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL14494879 0.77 CHRM2 (0.46) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL13180255 0.77 CHRM2 (0.59) CHRM2CHRM3CHRM1SIGMAR1CHRM4
SCHEMBL13145763 0.77 CHRM2 (0.46) CHRM2CHRM3CHRM1SIGMAR1CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240026358-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS THEREOF WAVE LIFE SCIENCES LTD. (SG) 2024-01-25 US disclosed
US-20230339902-A1 TRICYCLIC LIGANDS FOR DEGRADATION OF IKZF2 OR IKZF4 C4 THERAPEUTICS, INC. (US) 2023-10-26 US disclosed
WO-2023144793-A1 POL THETA INHIBITORS RHIZEN PHARMACEUTICALS AG (CH) 2023-08-03 WO disclosed
WO-2023091644-A2 HSD17B13-RELATED DOUBLE STRANDED OLIGONUCLEOTIDE COMPOSITIONS AND METHODS RELATING THERETO WAVE LIFE SCIENCES LTD. (SG) 2023-05-25 WO disclosed
WO-2023049218-A1 DOUBLE STRANDED OLIGONUCLEOTIDE COMPOSITIONS AND METHODS RELATING THERETO WAVE LIFE SCIENCES LTD. (SG) 2023-03-30 WO disclosed
WO-2022099159-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS THEREOF WAVE LIFE SCIENCES LTD. (SG) 2022-05-12 WO disclosed
WO-2022081925-A1 TRICYCLIC LIGANDS FOR DEGRADATION OF IKZF2 OR IKZF4 C4 THERAPEUTICS, INC. (US) 2022-04-21 WO disclosed
US-10017488-B2 3-substituted carbonyl-naphtho[2,3-B]furane derivative or pharmaceutically acceptable salt thereof BOSTON BIOMEDICAL, INC. (US) 2018-07-10 US disclosed
US-10017488-B2 3-substituted carbonyl-naphtho[2,3-B]furane derivative or pharmaceutically acceptable salt thereof BOSTON BIOMEDICAL, INC. (US) 2018-07-10 US disclosed
US-20170174646-A1 3-SUBSTITUTED CARBONYL-NAPHTHO[2,3-B]FURANE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF BOSTON BIOMEDICAL, INC. (US) 2017-06-22 US disclosed
US-20170174646-A1 3-SUBSTITUTED CARBONYL-NAPHTHO[2,3-B]FURANE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF BOSTON BIOMEDICAL, INC. (US) 2017-06-22 US disclosed
WO-2015120304-A1 3-SUBSTITUTED CARBONYL-NAPHTHO[2,3-B]FURANE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF BOSTON BIOMEDICAL, INC. (US) 2015-08-13 WO disclosed
WO-2009147476-A1 NOVEL PDE INHIBITORS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-12-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230339902-A1 TRICYCLIC LIGANDS FOR DEGRADATION OF IKZF2 OR IKZF4 IKZF1, IKZF3, IKZF2 CHRM2 4704/4885CHRM3 4601/4885CHRM1 4726/4885
US-20170174646-A1 3-SUBSTITUTED CARBONYL-NAPHTHO[2,3-B]FURANE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF FGFR3, FGFR1, FGF2 CHRM2 4064/4885CHRM3 4255/4885CHRM1 3262/4885
US-10017488-B2 3-substituted carbonyl-naphtho[2,3-B]furane derivative or pharmaceutically acceptable salt thereof FGFR3, FGFR1, FGF2 CHRM2 4064/4885CHRM3 4255/4885CHRM1 3262/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.